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PM376 Direct phosphorylation of the human cardiac L-type calcium channel alpha subunit by cAMP-dependent protein kinase alters function
Journal article   Peer reviewed

PM376 Direct phosphorylation of the human cardiac L-type calcium channel alpha subunit by cAMP-dependent protein kinase alters function

Henrietta Cserne Szappanos, David Longman, Tanzila Mahzabin, Padmapriya Muralidharan, Evan Ingley and Livia Hool
Global heart, Vol.9(1), p.e137
2014

Abstract

The L-type calcium channel plays a critical role in excitation-contraction coupling by mediating calcium influx into cardiomyocytes. In vivo, beta-adrenergic receptor stimulation is proposed to increase the activity of the channel via cAMP-dependent protein kinase A (PKA) phosphorylation. It is not clear whether direct phosphorylation of the channel protein is sufficient to alter function. In addition, while several consensus phosphorylation sites exist, the site/s responsible for increased channel activity remains unknown.

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